SCHEMBL6283602

SCHEMBL6283602

COc1cccc(C([O])[N+](=O)[O-])c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 1/20 0.47
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
CNR1 P21554 1/20 0.43
AOC3 Q16853 3/20 0.43
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
ACHE P22303 1/20 0.41
CASR P41180 2/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27656326 0.84 FBP1 (0.49) FBP1MAPK1L3MBTL1CHRM2CHRM1
SCHEMBL267537 0.83 MAPK1 (0.49) FBP1MAPK1L3MBTL1CHRM2CHRM1
SCHEMBL3826149 0.79 L3MBTL1 (0.49) FBP1MAPK1L3MBTL1CHRM2CHRM1
SCHEMBL6280529 0.78 FBP1 (0.46) FBP1MAPK1L3MBTL1GAAKMT2A
SCHEMBL20514192 0.78 MAPK1 (0.51) FBP1MAPK1L3MBTL1CHRM2CHRM1
SCHEMBL19169780 0.78 MAPK1 (0.51) FBP1MAPK1L3MBTL1CHRM2CHRM1
Hydrochloric Acid SCHEMBL11120361 0.78 MAPK1 (0.46) FBP1MAPK1L3MBTL1CHRM2CHRM1
SCHEMBL2093766 0.77 L3MBTL1 (0.53) L3MBTL1CHRM2CHRM1CHRM3AOC3
SCHEMBL7455624 0.76 MAPK1 (0.59) FBP1MAPK1L3MBTL1CHRM2CHRM1
SCHEMBL6204864 0.76 L3MBTL1 (0.51) L3MBTL1CHRM2CHRM1CHRM3AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP claimed
JP-2000502332-A 2000-02-29 JP claimed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP claimed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO claimed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO claimed
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed