SCHEMBL6284453

SCHEMBL6284453

COc1ccc(-c2nc(C(F)F)oc2-c2ccc(OC(C)O)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 7/20 0.36
KDM4E B2RXH2 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
IKBKB O14920 1/20 0.34
DHFR P00374 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 2/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6539500 0.86 ESR2 (0.47) PPARDKDM4EALDH1A1LMNATP53
SCHEMBL6230071 0.86 ESR2 (0.47) PPARDKDM4EALDH1A1LMNATP53
SCHEMBL13352330 0.83 CYP11B1 (0.42) PPARDKDM4ETDP1ALDH1A1LMNA
SCHEMBL6229912 0.81 PPARD (0.40) PPARDKDM4EALDH1A1IKBKBHPGD
SCHEMBL6538959 0.81 PPARD (0.40) PPARDKDM4EALDH1A1IKBKBHPGD
SCHEMBL6539133 0.81 PTGS2 (0.43) PPARDHDAC6
SCHEMBL6229835 0.80 KMT2A (0.39) PPARDKDM4EALDH1A1HPGDMAPT
SCHEMBL6538578 0.79 PPARD (0.54) PPARDKDM4EALDH1A1
SCHEMBL6538981 0.78 MAOB (0.54) PPARDKDM4EALDH1A1TP53HPGD
SCHEMBL6539783 0.78 ALDH1A1 (0.39) PPARDKDM4EALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583749-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE Astellas Pharma Inc. (JP) 2005-10-12 EP claimed
WO-2004065374-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE ASTELLAS PHARMA INC. (JP) 2004-08-05 WO claimed