SCHEMBL6286214

SCHEMBL6286214

O=c1c2ccccc2[nH]c(=S)n1-c1cccc(Cl)c1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 3/20 0.62
PDE7B Q9NP56 1/20 0.62
NPSR1 Q6W5P4 3/20 0.59
ALOX12 P18054 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
HPGD P15428 1/20 0.59
HTT P42858 3/20 0.58
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
MAPT P10636 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
RXFP1 Q9HBX9 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6280728 0.81 PDE7A (0.63) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL10550539 0.80 HTT (0.76) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL21436060 0.78 ALOX12 (0.70) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL6282188 0.78 PDE7A (0.63) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL18239972 0.78 HTT (0.67) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL6283505 0.78 PDE7A (0.77) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL30103233 0.77 PDE7A (1.00) PDE7APDE7BNPSR1MEN1KMT2A
SCHEMBL844588 0.77 PDE7A (1.00) PDE7APDE7BNPSR1MEN1KMT2A
SCHEMBL6284203 0.77 PDE7A (0.61) PDE7APDE7BNPSR1ALOX12MEN1
SCHEMBL6981997 0.75 KDM4E (0.74) PDE7APDE7BNPSR1ALOX12MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996020178-A1 NOVEL HETEROCYCLES AS CHOLECYSTOKININ (CCK) LIGANDS WARNER-LAMBERT COMPANY (US) 1996-07-04 WO claimed
US-6897213-B1 Heterocycles as cholecystokinin (CCK) ligands WARNER-LAMBERT COMPANY (US) 2005-05-24 US disclosed
WO-1996020178-A1 NOVEL HETEROCYCLES AS CHOLECYSTOKININ (CCK) LIGANDS WARNER-LAMBERT COMPANY (US) 1996-07-04 WO disclosed