SCHEMBL6287945

SCHEMBL6287945

COC(=O)Cc1c(C)[nH]c2cc(C(F)(F)F)ccc12

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.48
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
MAPT P10636 1/20 0.47
MCL1 Q07820 3/20 0.46
AKR1C3 P42330 1/20 0.44
EGFR P00533 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
AKR1C2 P52895 1/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6290568 0.85 KDM4E (0.58) KIF11TMEM97SIGMAR1MAPTMCL1
SCHEMBL6282260 0.82 MAPT (0.55) KIF11MAPTEGFRMEN1KMT2A
SCHEMBL8292165 0.80 MCL1 (0.47) MAPTMCL1EGFRMEN1KMT2A
SCHEMBL13299834 0.79 AKR1C2 (0.41) MAPTAKR1C3EGFRMEN1KMT2A
SCHEMBL11328478 0.79 MEN1 (0.48) KIF11MAPTMEN1KMT2AAKR1C2
SCHEMBL27532185 0.78 PTGS2 (0.61) MCL1AKR1C3
SCHEMBL12255237 0.78 MTNR1A (0.46) MAPTAKR1C3EGFRMEN1KMT2A
SCHEMBL28631063 0.78 MEN1 (0.50) KIF11MAPTEGFRMEN1KMT2A
SCHEMBL1191332 0.76 KDM4E (0.69) MAPTEGFRAKR1C2
SCHEMBL14487672 0.75 MEN1 (0.50) KIF11MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6887890-B2 Compounds exhibiting thrombopoietin-like activities CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2005-05-03 US disclosed
US-20030162724-A1 Compounds exhibiting thrombopoietin-like activities CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-08-28 US disclosed
EP-1291341-A1 COMPOUNDS EXHIBITING THROMBOPOIETIN-LIKE ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162724-A1 Compounds exhibiting thrombopoietin-like activities MPL, THPO, TEK KIF11 4720/4885TMEM97 1605/4885SIGMAR1 1216/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.