SCHEMBL6289952

SCHEMBL6289952

N#Cc1ccc(Oc2cccc(CN)c2)cc1C#N

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.54
MAOB P27338 6/20 0.53
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
AR P10275 3/20 0.44
ST14 Q9Y5Y6 1/20 0.44
MAOA P21397 3/20 0.43
NPSR1 Q6W5P4 1/20 0.42
PDE4B Q07343 1/20 0.41
F10 P00742 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19280735 0.84 CYP19A1 (0.54) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL6289949 0.84 CYP19A1 (0.54) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL16310207 0.84 CYP19A1 (0.54) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL9746473 0.83 CYP19A1 (0.52) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL9746014 0.83 CYP19A1 (0.52) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL1374021 0.83 CYP19A1 (0.67) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL31168160 0.83 CYP19A1 (0.67) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL5145150 0.83 CYP19A1 (0.67) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL13908822 0.81 CYP19A1 (0.65) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL4949955 0.81 ST14 (0.58) MAOBALDH1A1ST14F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6867200-B1 (Hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-15 US disclosed