SCHEMBL6289949

SCHEMBL6289949

N#Cc1ccc(Oc2cccc(C[NH])c2)cc1C#N

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.54
MAOB P27338 6/20 0.53
ALDH1A1 P00352 3/20 0.45
HPGD P15428 2/20 0.45
AR P10275 4/20 0.44
MAOA P21397 4/20 0.43
NPSR1 Q6W5P4 1/20 0.42
PDE4B Q07343 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
PGGT1B P53609 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16310207 0.84 CYP19A1 (0.54) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL6289952 0.84 CYP19A1 (0.54) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL19280735 0.84 CYP19A1 (0.54) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL9746473 0.83 CYP19A1 (0.52) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL9746014 0.83 CYP19A1 (0.52) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL1374021 0.83 CYP19A1 (0.67) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL31168160 0.83 CYP19A1 (0.67) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL5145150 0.83 CYP19A1 (0.67) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL13908822 0.81 CYP19A1 (0.65) CYP19A1MAOBALDH1A1HPGDAR
SCHEMBL4581525 0.79 CYP19A1 (0.65) CYP19A1MAOBALDH1A1HPGDAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6867200-B1 (Hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-15 US disclosed