SCHEMBL6296969

SCHEMBL6296969

O=S(=O)(Nc1ccc(O)cc1)c1ccc(-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UQCRB P14927 3/20 1.00
MEN1 O00255 3/20 0.65
KMT2A Q03164 3/20 0.65
ALDH1A1 P00352 1/20 0.65
PKM P14618 1/20 0.65
MAPT P10636 3/20 0.61
GAA P10253 2/20 0.61
HTT P42858 2/20 0.61
MAPK1 P28482 1/20 0.61
RECQL P46063 1/20 0.61
HDAC1 Q13547 3/20 0.59
HDAC3 O15379 2/20 0.59
HDAC4 P56524 2/20 0.59
HDAC7 Q8WUI4 2/20 0.59
HDAC2 Q92769 2/20 0.59
HDAC10 Q969S8 2/20 0.59
HDAC11 Q96DB2 2/20 0.59
HDAC8 Q9BY41 2/20 0.59
HDAC6 Q9UBN7 2/20 0.59
HDAC9 Q9UKV0 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21086838 0.93 UQCRB (0.86) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL930801 0.89 UQCRB (0.80) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL523563 0.89 UQCRB (0.80) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL27428246 0.87 UQCRB (0.77) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL28178888 0.87 UQCRB (0.77) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL812677 0.87 KMT2A (0.77) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL13480185 0.87 KMT2A (0.77) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL1592323 0.87 UQCRB (0.76) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL13167612 0.85 KMT2A (0.80) UQCRBMEN1KMT2AALDH1A1PKM
SCHEMBL7824383 0.84 UQCRB (0.72) UQCRBMEN1KMT2AALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114751863-B Terpastacin derivative, preparation method thereof and application thereof in preparation of hypoxia factor inhibitor 中国科学院南海海洋研究所 2024-01-05 CN disclosed
CN-115634224-A Application of Terestacin derivative in preparation of medicine for treating brain glioma 中国科学院南海海洋研究所 2023-01-24 CN disclosed
CN-114751863-A Terestacin derivative, preparation method thereof and application of Terestacin derivative in preparation of low-oxygen factor inhibitor 中国科学院南海海洋研究所 2022-07-15 CN disclosed
US-9371286-B2 Pharmaceutical composition with enhanced efficacy for inhibiting angiogenesis INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2016-06-21 US disclosed
US-9371286-B2 Pharmaceutical composition with enhanced efficacy for inhibiting angiogenesis INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2016-06-21 US disclosed
US-20140315947-A1 PHARMACEUTICAL COMPOSITION WITH ENHANCED EFFICACY FOR INHIBITING ANGIOGENESIS INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2014-10-23 US disclosed
US-20140315947-A1 PHARMACEUTICAL COMPOSITION WITH ENHANCED EFFICACY FOR INHIBITING ANGIOGENESIS INDUSTRY-ACADEMIC COOPERATION FOUNDATION, YONSEI UNIVERSITY (KR) 2014-10-23 US disclosed
US-6921740-B1 Electron-receiving compound and thermal recording material MITSUBISHI PAPER MIILS LTD. (JP) 2005-07-26 US disclosed
US-6579829-B2 Aromatic sulfonamide compound MITSUI CHEMICALS, INC. (JP) 2003-06-17 US disclosed
EP-1138517-A2 Developer composition and heat sensitive recording material Mitsui Chemicals, Inc. (JP) 2001-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140315947-A1 PHARMACEUTICAL COMPOSITION WITH ENHANCED EFFICACY FOR INHIBITING ANGIOGENESIS UQCRB, UQCRC1, UQCRC2 UQCRB 1/4885MEN1 4790/4885KMT2A 4308/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.