SCHEMBL6299339

SCHEMBL6299339

CC(C)=CC(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.71
ALDH1A1 P00352 3/20 0.71
SMN1; SMN2 Q16637 2/20 0.55
TSHR P16473 1/20 0.55
CASP1 P29466 1/20 0.55
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPK1 P28482 1/20 0.50
HIF1A Q16665 1/20 0.50
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
GABRA1 P14867 6/20 0.49
GABRG2 P18507 6/20 0.49
GABRB3 P28472 6/20 0.49
GABRB2 P47870 4/20 0.49
GABRB1 P18505 2/20 0.49
KDM4E B2RXH2 1/20 0.49
POLB P06746 2/20 0.46
THRB P10828 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11231466 0.87 ALDH1A1 (0.69) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL11231463 0.87 ALDH1A1 (0.69) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL10999586 0.83 ALDH1A1 (0.63) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL6299219 0.82 MAPT (0.61) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL3310055 0.80 ALDH1A1 (0.59) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL3310049 0.80 ALDH1A1 (0.59) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL3310052 0.80 ALDH1A1 (0.59) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL30513965 0.79 SMN1; SMN2 (0.61) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL1697502 0.79 SMN1; SMN2 (0.61) MAPTALDH1A1SMN1; SMN2TSHRCASP1
SCHEMBL322161 0.78 TSHR (0.65) MAPTALDH1A1SMN1; SMN2TSHRCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911469-B2 Sulfonamide compounds and pharmaceutical use thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-28 US disclosed
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2002-07-25 US disclosed
US-6348474-B1 COMPOUNDS AS ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-0995742-A1 SULFONAMIDE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity PDE2A, PDE3A, PDE12 MAPT 4591/4885ALDH1A1 570/4885SMN1; SMN2 186/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.