SCHEMBL6299366

SCHEMBL6299366

Cc1oc2ccc(C(=O)NS(=O)(=O)/C=C/c3ccccc3)cc2c1Cc1ccc(Cl)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
SLC26A4 O43511 1/20 0.40
POLB P06746 1/20 0.40
BCAT1 P54687 5/20 0.39
TBXA2R P21731 1/20 0.37
PTGFR P43088 1/20 0.37
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
PTGIR P43119 1/20 0.37
PTGDR Q13258 1/20 0.37
HDAC8 Q9BY41 3/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PPARG P37231 1/20 0.36
KMT2A Q03164 1/20 0.35
EGFR P00533 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 2/20 0.34
TTR P02766 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6299371 1.00 ALDH1A1 (0.40) ALDH1A1SLC26A4POLBBCAT1TBXA2R
SCHEMBL6135003 0.91 SCN9A (0.36) BCAT1HDAC8HDAC6KMT2A
SCHEMBL6298789 0.91 ALDH1A1 (0.35) ALDH1A1BCAT1KMT2AKDM4EHTT
SCHEMBL6135001 0.91 SCN9A (0.36) BCAT1HDAC8HDAC6KMT2A
SCHEMBL6298792 0.91 ALDH1A1 (0.35) ALDH1A1BCAT1KMT2AKDM4EHTT
SCHEMBL6299324 0.88 PPARG (0.40) SLC26A4POLBBCAT1TBXA2RPTGFR
SCHEMBL6299326 0.88 PPARG (0.40) SLC26A4POLBBCAT1TBXA2RPTGFR
SCHEMBL6301261 0.87 FLT1 (0.47) SLC26A4POLBBCAT1
SCHEMBL5882071 0.83 MAPT (0.42) ALDH1A1TBXA2RPTGFRPTGER3PTGER2
SCHEMBL5882069 0.83 MAPT (0.42) ALDH1A1TBXA2RPTGFRPTGER3PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911469-B2 Sulfonamide compounds and pharmaceutical use thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-28 US disclosed
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-09-16 US disclosed
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2002-07-25 US disclosed
US-6348474-B1 COMPOUNDS AS ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-0995742-A1 SULFONAMIDE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity PDE2A, PDE3A, PDE12 ALDH1A1 570/4885SLC26A4 2801/4885POLB 2385/4885
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications PDE2A, PDE3A, PYGM ALDH1A1 1067/4885SLC26A4 3789/4885POLB 1050/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.