SCHEMBL6300596

SCHEMBL6300596

O=C1C(Br)Cc2ccccc2CC1Br

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
ANPEP P15144 1/20 0.42
IDO1 P14902 3/20 0.39
CYP2A6 P11509 1/20 0.39
ACHE P22303 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PLAU P00749 1/20 0.37
CYP19A1 P11511 1/20 0.36
ADRA2A P08913 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL296403 0.75 ACHE (0.59) ACHECYP19A1CES1
SCHEMBL29752636 0.75 ACHE (0.59) ACHECYP19A1CES1
SCHEMBL1923692 0.73 IDO1 (0.46) ANPEPIDO1CA1CA2PLAU
SCHEMBL31490422 0.73 IDO1 (0.46) ANPEPIDO1CA1CA2PLAU
SCHEMBL11822112 0.72 HTR2A (0.57) ANPEP
SCHEMBL1170559 0.72
SCHEMBL3345089 0.70 MAOB (0.43) CYP1A2ACHECYP19A1
SCHEMBL2485525 0.70 IDO1 (0.44) CYP1A2ANPEPIDO1ACHECA1
SCHEMBL13866808 0.70 IDO1 (0.44) CYP1A2ANPEPIDO1ACHECA1
SCHEMBL6317426 0.70 IDO1 (0.44) CYP1A2ANPEPIDO1ACHECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6846833-B2 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same LES LABORATORIES SERVIER (FR) 2005-01-25 US disclosed
EP-1268429-B1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2004-08-18 EP disclosed
EP-1268429-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME Les Laboratoires Servier (FR) 2003-01-02 EP disclosed
WO-2001079172-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER Departament Brevets/Fontanes (FR) 2001-10-25 WO disclosed