SCHEMBL6300831

SCHEMBL6300831

CCOc1ccc(C(=O)N(CC(=O)N2CCN(C3CCN(C)CC3)CC2)c2ccccc2C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.45
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
SLC6A5 Q9Y345 4/20 0.42
GAA P10253 1/20 0.40
NPC1 O15118 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
L3MBTL3 Q96JM7 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ORAI1 Q96D31 1/20 0.38
RBP4 P02753 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4842608 0.92 KDM4E (0.43) ACHEKEAP1NFE2L2SLC6A5L3MBTL1
Hydrochloric Acid SCHEMBL4841723 0.91 KDM4E (0.42) ACHEKEAP1NFE2L2SLC6A5L3MBTL1
Hydrochloric Acid SCHEMBL4832567 0.91 KDM4E (0.42) ACHEKEAP1NFE2L2SLC6A5L3MBTL1
SCHEMBL4832702 0.81 GAA (0.41) ACHEKEAP1NFE2L2GAAL3MBTL1
Hydrochloric Acid SCHEMBL4832297 0.81 F10 (0.50) L3MBTL1L3MBTL3KDM4EALDH1A1
SCHEMBL6379660 0.80 ACHE (0.48) ACHESLC6A5GAAGPR119L3MBTL1
SCHEMBL4840253 0.78 KDM4E (0.45) ACHEL3MBTL1L3MBTL3KDM4EALDH1A1
Hydrochloric Acid SCHEMBL4841921 0.78 KDM4E (0.44) ACHEKEAP1NFE2L2L3MBTL1L3MBTL3
SCHEMBL4832817 0.77 ALDH1A1 (0.44) ACHEL3MBTL1L3MBTL3KDM4EALDH1A1
Hydrochloric Acid SCHEMBL4840498 0.76 ALDH1A1 (0.43) ACHEL3MBTL1L3MBTL3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936611-B2 Serine protease inhibitors ELI LILLY AND COMPANY (US) 2005-08-30 US claimed