SCHEMBL6301285

SCHEMBL6301285

Cc1cc(C(=O)NS(=O)(=O)/C=C/c2ccccc2)nc2c1nc(C)n2Cc1ccc(-c2ccc(Cl)s2)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.34
AGTR2 P50052 1/20 0.34
PPARG P37231 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
HSD17B13 Q7Z5P4 1/20 0.32
PIK3CB P42338 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6301292 1.00 AGTR1 (0.34) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6300758 0.90 PTGER3 (0.34) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6305101 0.90 PTGER3 (0.34) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6300462 0.89 PPARG (0.39) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6300461 0.89 PPARG (0.39) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6298724 0.86 PPARG (0.36) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6298722 0.86 PPARG (0.36) AGTR1AGTR2PPARGALDH1A1MAPT
SCHEMBL6298974 0.83 MEN1 (0.38) PPARGALDH1A1
SCHEMBL6298981 0.83 MEN1 (0.38) PPARGALDH1A1
SCHEMBL6305971 0.83 PPARG (0.49) AGTR1AGTR2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911469-B2 Sulfonamide compounds and pharmaceutical use thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-28 US disclosed
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-09-16 US disclosed
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2002-07-25 US disclosed
EP-0995742-A1 SULFONAMIDE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity PDE2A, PDE3A, PDE12 AGTR1 58/4885AGTR2 48/4885PPARG 2713/4885
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications PDE2A, PDE3A, PYGM AGTR1 269/4885AGTR2 127/4885PPARG 1366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.