SCHEMBL6301756

SCHEMBL6301756

N#Cc1cccc(CNc2ccccn2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP1 P07148 1/20 0.61
FABP6 P51161 1/20 0.61
CXCR4 P61073 1/20 0.58
CYP1A2 P05177 7/20 0.56
CYP2C19 P33261 7/20 0.56
CLK4 Q9HAZ1 6/20 0.56
CYP3A4 P08684 5/20 0.56
CYP2D6 P10635 4/20 0.56
LMNA P02545 2/20 0.56
HSD17B10 Q99714 5/20 0.54
ALDH1A1 P00352 5/20 0.54
MAPK1 P28482 3/20 0.54
USP2 O75604 2/20 0.54
VNN1 O95497 3/20 0.53
TSHR P16473 4/20 0.52
ALOX15 P16050 2/20 0.52
TP53 P04637 2/20 0.52
CYP2C9 P11712 2/20 0.52
KDM4E B2RXH2 3/20 0.51
GABRG2 P18507 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10054969 0.84 FABP1 (0.79) FABP1FABP6CXCR4CYP1A2CYP2C19
SCHEMBL29580004 0.83 CXCR4 (0.74) FABP1FABP6CXCR4CYP1A2CYP2C19
SCHEMBL5879525 0.83 CXCR4 (0.74) FABP1FABP6CXCR4CYP1A2CYP2C19
SCHEMBL2194571 0.77 KDM5A (0.61) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL2230559 0.77 FABP1 (1.00) FABP1FABP6CXCR4CYP1A2CYP2D6
SCHEMBL29664808 0.77 FABP1 (1.00) FABP1FABP6CXCR4CYP1A2CYP2D6
SCHEMBL23938199 0.77 KDM4E (0.69) FABP1FABP6CXCR4TSHRTP53
SCHEMBL11573094 0.77 FABP1 (0.67) FABP1FABP6CXCR4CYP1A2CYP2C19
SCHEMBL4718827 0.77 FABP1 (0.67) FABP1FABP6CXCR4ALDH1A1TSHR
SCHEMBL6301782 0.77 FABP1 (0.67) FABP1FABP6CXCR4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113651811-B Isoxazole-containing pyridopyrimidone compound and preparation method and application thereof 贵州大学 2022-06-07 CN disclosed
US-6846833-B2 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same LES LABORATORIES SERVIER (FR) 2005-01-25 US disclosed
EP-1268429-B1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2004-08-18 EP disclosed
EP-1268429-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME Les Laboratoires Servier (FR) 2003-01-02 EP disclosed
WO-2001079172-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER Departament Brevets/Fontanes (FR) 2001-10-25 WO disclosed