SCHEMBL6307014

SCHEMBL6307014

COc1ccc(-c2nc3ccc(OC)cc3c(=O)n2CCCN)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F11 P03951 3/20 0.67
ALDH1A1 P00352 6/20 0.55
MAPK1 P28482 3/20 0.55
TSHR P16473 1/20 0.55
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HPGD P15428 4/20 0.53
KDM4E B2RXH2 3/20 0.53
MAPT P10636 3/20 0.53
LMNA P02545 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.52
POLB P06746 2/20 0.50
RXFP1 Q9HBX9 2/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
HTR1A P08908 1/20 0.48
DYRK3 O43781 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6308394 0.95 F11 (0.65) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6308567 0.94 F11 (0.64) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6306921 0.94 F11 (0.63) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6314809 0.93 F11 (0.63) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6306850 0.93 F11 (0.59) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6306796 0.92 F11 (0.61) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6308080 0.91 F11 (0.57) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6306810 0.91 F11 (0.62) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6308495 0.90 F11 (0.59) F11ALDH1A1MAPK1TSHRMEN1
SCHEMBL6307622 0.90 F11 (0.59) F11ALDH1A1MAPK1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed