SCHEMBL6314809

SCHEMBL6314809

COc1cc(OC)cc(-c2ccc(-c3nc4ccc(OC)cc4c(=O)n3CCCN)cc2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F11 P03951 1/20 0.63
ALDH1A1 P00352 6/20 0.49
MAPK1 P28482 3/20 0.49
RXFP1 Q9HBX9 2/20 0.49
TSHR P16473 1/20 0.49
POLB P06746 1/20 0.49
HPGD P15428 4/20 0.47
MAPT P10636 4/20 0.47
KDM4E B2RXH2 3/20 0.47
LMNA P02545 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
ADRB2 P07550 1/20 0.45
ADRB1 P08588 1/20 0.45
HTR1A P08908 1/20 0.45
AVPR1B P47901 2/20 0.44
DYRK3 O43781 1/20 0.44
CLK1 P49759 1/20 0.44
CLK2 P49760 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307014 0.93 F11 (0.67) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6307757 0.93 F11 (0.54) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6308567 0.93 F11 (0.64) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6308394 0.91 F11 (0.65) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6315037 0.91 POLB (0.54) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6306921 0.90 F11 (0.63) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6309730 0.89 ALDH1A1 (0.59) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6308835 0.88 F11 (0.58) F11ALDH1A1RXFP1POLBAVPR1B
SCHEMBL6306796 0.88 F11 (0.61) F11ALDH1A1MAPK1RXFP1TSHR
SCHEMBL6306850 0.87 F11 (0.59) F11ALDH1A1MAPK1RXFP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed