SCHEMBL6307025

SCHEMBL6307025

COc1ccc2nc(/C=C/c3ccc(N(C)C)cc3)n(Cc3cccc(CN)c3)c(=O)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 8/20 0.46
TP53 P04637 2/20 0.46
HPGD P15428 3/20 0.44
MAPT P10636 3/20 0.44
NPC1 O15118 2/20 0.44
LMNA P02545 2/20 0.44
NFKB1 P19838 2/20 0.44
HTT P42858 2/20 0.44
RAB9A P51151 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
GLA P06280 2/20 0.43
GAA P10253 1/20 0.43
NPY1R P25929 1/20 0.43
NPY2R P49146 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307031 1.00 MEN1 (0.49) MEN1KMT2AALDH1A1TP53HPGD
SCHEMBL6313198 0.91 ALDH1A1 (0.55) KMT2AALDH1A1TP53HPGDMAPT
SCHEMBL6313191 0.91 ALDH1A1 (0.55) KMT2AALDH1A1TP53HPGDMAPT
SCHEMBL7554195 0.89 ALDH1A1 (0.55) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL7554190 0.89 ALDH1A1 (0.55) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL6313858 0.88 KMT2A (0.51) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL6313851 0.88 KMT2A (0.51) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL6309743 0.87 KMT2A (0.64) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL6309745 0.87 KMT2A (0.64) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL6307872 0.84 ALDH1A1 (0.46) MEN1KMT2AALDH1A1TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed