SCHEMBL6307495

SCHEMBL6307495

NC(=O)C(Cc1ccccc1)N1C(=O)c2ccc(OCc3ccc(F)cc3)cc2C1=O

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.60
L3MBTL1 Q9Y468 3/20 0.60
ALDH1A1 P00352 2/20 0.60
GAA P10253 1/20 0.50
KMT2A Q03164 4/20 0.49
GPR34 Q9UPC5 2/20 0.48
AADAT Q8N5Z0 1/20 0.46
MEN1 O00255 3/20 0.46
CYP2D6 P10635 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
NR4A2 P43354 1/20 0.44
MAOB P27338 1/20 0.44
PARP10 Q53GL7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307483 1.00 POLB (0.60) POLBL3MBTL1ALDH1A1GAAKMT2A
SCHEMBL3505013 0.87 MAOB (0.47) POLBL3MBTL1ALDH1A1KMT2AMEN1
SCHEMBL3505017 0.87 MAOB (0.47) POLBL3MBTL1ALDH1A1KMT2AMEN1
SCHEMBL4467004 0.87 POLB (0.76) POLBL3MBTL1ALDH1A1GAAKMT2A
SCHEMBL13919525 0.87 POLB (0.76) POLBL3MBTL1ALDH1A1GAAKMT2A
SCHEMBL6309095 0.86 MAOB (0.46) L3MBTL1KMT2AMEN1NR4A2MAOB
SCHEMBL5823994 0.86 MAOB (0.46) POLBL3MBTL1ALDH1A1KMT2AMEN1
SCHEMBL5618422 0.86 MAOB (0.46) POLBL3MBTL1ALDH1A1KMT2AMEN1
SCHEMBL6309098 0.86 MAOB (0.46) L3MBTL1KMT2AMEN1NR4A2MAOB
SCHEMBL6309099 0.86 MAOB (0.46) L3MBTL1KMT2AMEN1NR4A2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1277820-C Phthalimido derivatives as inhibitors of monoamine oxidase B HOFFMANN LA ROCHE (CH) 2006-10-04 CN disclosed
CN-1642911-A Phthalimido derivatives as inhibitors of monoamine oxidase B HOFFMANN LA ROCHE (CH) 2005-07-20 CN disclosed
US-6903095-B2 Nitrogen compounds such as 2-(5-(4-Fluoro-benzyloxy)-1,3-dioxo -1,3-dihydro-isoindol-2-yl)-acetamide, used for prophylaxis of Alzheimer's disease; amine oxidase inhibitors HOFFMANN-LA ROCHE INC. (US) 2005-06-07 US disclosed
US-20040229871-A1 Phthalimido derivatives and a process for their preparation CESURA ANDREA (CH) 2004-11-18 US disclosed
US-6660736-B2 MAO-B inhibitors HOFFMANN-LA ROCHE INC. 2003-12-09 US disclosed
US-20030195208-A1 PHTHALIMIDO DERIVATIVES AND A PROCESS FOR THEIR PREPARATION HOFFMANN-LA ROCHE INC. 2003-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030195208-A1 PHTHALIMIDO DERIVATIVES AND A PROCESS FOR THEIR PREPARATION MAOB, MAOA, CYP4B1 POLB 568/4885L3MBTL1 2932/4885ALDH1A1 225/4885
US-20040229871-A1 Phthalimido derivatives and a process for their preparation MAOB, MAOA, CYP4B1 POLB 568/4885L3MBTL1 2932/4885ALDH1A1 225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.