SCHEMBL6314905

SCHEMBL6314905

CCN(CC)CCn1c(-c2ccc(C)cc2)nc2ccccc2c1=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.64
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
CASR P41180 1/20 0.56
RXFP1 Q9HBX9 2/20 0.56
TOP2A P11388 1/20 0.54
SMN1; SMN2 Q16637 4/20 0.53
ABCC1 P33527 1/20 0.53
RAB9A P51151 2/20 0.52
LMNA P02545 1/20 0.52
RECQL P46063 1/20 0.52
TSHR P16473 2/20 0.52
GAA P10253 2/20 0.51
NPC1 O15118 1/20 0.51
POLB P06746 1/20 0.51
RAD52 P43351 1/20 0.51
SMARCA2 P51531 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550755 0.94 CASR (0.64) ALDH1A1MEN1KMT2ACASRTOP2A
SCHEMBL6308150 0.88 ALDH1A1 (0.67) ALDH1A1MEN1KMT2ACASRRXFP1
SCHEMBL6306907 0.84 MEN1 (0.59) ALDH1A1MEN1KMT2ACASRRXFP1
SCHEMBL6313235 0.82 ALDH1A1 (0.70) ALDH1A1MEN1KMT2ACASRRXFP1
SCHEMBL6308959 0.81 ABCC1 (0.47) ALDH1A1MEN1KMT2ARXFP1TOP2A
SCHEMBL5921364 0.81 CASR (0.85) ALDH1A1MEN1KMT2ACASRRXFP1
SCHEMBL6313584 0.81 CASR (0.67) ALDH1A1MEN1KMT2ACASRTOP2A
SCHEMBL6308206 0.81 ALDH1A1 (0.64) ALDH1A1MEN1KMT2ACASRRXFP1
SCHEMBL6306022 0.80 EGFR (0.58) ALDH1A1MEN1KMT2ACASRRXFP1
SCHEMBL6314431 0.80 MEN1 (0.67) ALDH1A1MEN1KMT2ACASRRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed