SCHEMBL6320130

SCHEMBL6320130

Nc1onc(-c2ccc(Cl)s2)c1C(=O)NCc1ccccc1Br

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.55
CA2 P00918 3/20 0.55
CA4 P22748 3/20 0.55
CA7 P43166 3/20 0.55
ALDH1A1 P00352 2/20 0.46
PRNP P04156 1/20 0.42
KMT2A Q03164 2/20 0.42
P2RX7 Q99572 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 1/20 0.38
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6322701 0.90 CA1 (0.54) CA1CA2CA4CA7ALDH1A1
SCHEMBL6323533 0.90 ALDH1A1 (0.47) CA1CA2CA4CA7ALDH1A1
SCHEMBL6316785 0.88 CA1 (0.52) CA1CA2CA4CA7ALDH1A1
SCHEMBL6317667 0.88 CA2 (0.52) CA1CA2CA4CA7ALDH1A1
SCHEMBL6318552 0.87 ALDH1A1 (0.50) CA1CA2CA4CA7ALDH1A1
SCHEMBL6319063 0.86 CA2 (0.51) CA1CA2CA4CA7KMT2A
SCHEMBL6316598 0.85 CA1 (0.56) CA1CA2CA4CA7ALDH1A1
SCHEMBL6318170 0.84 ALDH1A1 (0.45) CA1CA2CA4CA7ALDH1A1
SCHEMBL6316464 0.81 HPGD (0.56) CA1CA2CA4CA7ALDH1A1
SCHEMBL6322551 0.80 CA1 (0.54) CA1CA2CA4CA7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050059657-A1 Aminoisoxazole derivatives active as kinase inhibitors PFIZER ITALIA S.R.L. (IT) 2005-03-17 US claimed
EP-1435948-A1 AMINOISOXAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS Pharmacia Italia S.p.A. (IT) 2004-07-14 EP claimed
WO-2003013517-A1 AMINOISOXAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS PHARMACIA ITALIA S.P.A. (IT) 2003-02-20 WO claimed
US-12420503-B2 Late-stage catalysis of fast room-temperature polymerizations ESSILOR INTERNATIONAL (FR) 2025-09-23 US disclosed
US-20250108574-A1 LATE-STAGE CATALYSIS OF FAST ROOM-TEMPERATURE POLYMERIZATIONS ESSILOR INTERNATIONAL (FR) 2025-04-03 US disclosed
EP-4253019-A1 LATE-STAGE CATALYSIS OF FAST ROOM-TEMPERATURE POLYMERIZATIONS Essilor International (FR) 2023-10-04 EP disclosed
US-20050059657-A1 Aminoisoxazole derivatives active as kinase inhibitors PFIZER ITALIA S.R.L. (IT) 2005-03-17 US disclosed
US-6844415-B1 Polymerizable compositions for making thio containing resins including a salt catalyst and process for making thio containing ESSILOR INTERNATIONAL-COMPAGNIE GENERAL D'OPTIQUE (FR) 2005-01-18 US disclosed
EP-1435948-A1 AMINOISOXAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS Pharmacia Italia S.p.A. (IT) 2004-07-14 EP disclosed
WO-2003013517-A1 AMINOISOXAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS PHARMACIA ITALIA S.P.A. (IT) 2003-02-20 WO disclosed
US-5973098-A CASTING OPTICAL LENSES ESSILOR INTERNATIONAL - COMPAGNIE GENERALE D'OPTIQUE (FR) 1999-10-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059657-A1 Aminoisoxazole derivatives active as kinase inhibitors MAP3K9, MAP3K19, MAP4K2 CA1 2406/4885CA2 2764/4885CA4 4029/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.