SCHEMBL6324844

SCHEMBL6324844

CC12CN(Cc3ccccc3)CC(C)(CN(C(=O)O)C1)C2O

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
TSHR P16473 3/20 0.48
CYP2D6 P10635 4/20 0.45
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 2/20 0.43
FUCA1 P04066 2/20 0.43
CYP3A4 P08684 2/20 0.42
HSD11B1 P28845 1/20 0.42
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6316162 0.89 GAA (0.57) GAAKMT2AMEN1TSHRALDH1A1
SCHEMBL6318216 0.84 GAA (0.45) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL20397168 0.81 GAA (0.46) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL6319658 0.79 GAA (0.54) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL20399590 0.79 DRD4 (0.44) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL20399589 0.79 DRD4 (0.44) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL29937252 0.73 GAA (0.47) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL29937256 0.73 GAA (0.47) GAAKMT2AMEN1TSHRCYP2D6
SCHEMBL2381838 0.72 CYP2D6 (0.67) KMT2AMEN1TSHRCYP2D6ALDH1A1
SCHEMBL6318884 0.71 S1PR5 (0.48) GAAKMT2AMEN1TSHRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6887881-B1 Bispidine compounds useful in the treatment of cardiac arrythmias ASTRAZENECA AB (SE) 2005-05-03 US disclosed
EP-1192154-B1 BISPIDINE COMPOUNDS USEFUL IN THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2004-03-17 EP disclosed