SCHEMBL6326778

SCHEMBL6326778

NC(=NCC(=O)O)c1ccc(O)c(CNc2ncnc3cc(C(=O)N4CCCC4)c(Cl)cc23)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 5/20 0.41
PDE5A O76074 3/20 0.36
CNR1 P21554 2/20 0.34
CNR2 P34972 1/20 0.34
AURKA O14965 3/20 0.33
RPS6KB1 P23443 3/20 0.33
AURKB Q96GD4 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPK1 P28482 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CSNK1D P48730 1/20 0.32
CSNK1G2 P78368 1/20 0.32
MAPK10 P53779 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311630 0.90 CDK1 (0.42) CDK1PDE5ACNR1CNR2AURKA
SCHEMBL8312247 0.88 CDK1 (0.39) CDK1PDE5ACNR1CNR2AURKA
SCHEMBL2995398 0.87 CDK1 (0.42) CDK1PDE5ACNR1CNR2AURKA
SCHEMBL6326818 0.82 CDK1 (0.47) CDK1PDE5ACNR1CNR2AURKA
SCHEMBL8308640 0.82 CDK1 (0.37) CDK1PDE5ACNR1CNR2ALDH1A1
Hydrochloric Acid SCHEMBL6322307 0.81 CDK1 (0.46) CDK1PDE5ACNR1CNR2AURKA
SCHEMBL6322214 0.81 CDK1 (0.39) CDK1PDE5ACNR1CNR2ALDH1A1
SCHEMBL8312292 0.79 CDK1 (0.36) CDK1PDE5AAURKARPS6KB1AURKB
SCHEMBL2991625 0.78 F10 (0.41) CDK1PDE5AAURKARPS6KB1AURKB
SCHEMBL6332101 0.78 CDK1 (0.39) CDK1PDE5AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597248-A2 SULFONAMIDE DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-11-23 EP disclosed
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed
WO-2004073606-A2 SULFONAMIDE DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2004-09-02 WO disclosed