SCHEMBL8312247

SCHEMBL8312247

N/C(=N\C(=O)c1ccccc1)c1ccc(O)c(CNc2ncnc3cc(C(=O)N4CCCC4)c(Cl)cc23)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.39
AURKA O14965 3/20 0.36
RPS6KB1 P23443 3/20 0.36
AURKB Q96GD4 2/20 0.36
PDE5A O76074 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
MAPK10 P53779 6/20 0.34
MAPK8 P45983 4/20 0.34
CSNK1D P48730 1/20 0.34
CSNK1G2 P78368 1/20 0.34
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.34
EGFR P00533 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312292 0.92 CDK1 (0.36) CDK1AURKARPS6KB1AURKBPDE5A
SCHEMBL8311630 0.88 CDK1 (0.42) CDK1AURKARPS6KB1AURKBPDE5A
SCHEMBL6326778 0.88 CDK1 (0.41) CDK1AURKARPS6KB1AURKBPDE5A
SCHEMBL2995398 0.86 CDK1 (0.42) CDK1AURKARPS6KB1AURKBPDE5A
SCHEMBL6322214 0.84 CDK1 (0.39) CDK1PDE5AKDM4EALDH1A1MAPK1
SCHEMBL8308640 0.83 CDK1 (0.37) CDK1PDE5AKDM4EALDH1A1MAPK1
SCHEMBL6326818 0.81 CDK1 (0.47) CDK1AURKARPS6KB1AURKBPDE5A
Hydrochloric Acid SCHEMBL6322307 0.80 CDK1 (0.46) CDK1AURKARPS6KB1AURKBPDE5A
SCHEMBL6324788 0.78 HPGD (0.41) CDK1AURKARPS6KB1AURKBPDE5A
SCHEMBL8308730 0.77 PDE5A (0.36) CDK1AURKARPS6KB1AURKBPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed