SCHEMBL8311630

SCHEMBL8311630

C/N=C(/N)c1ccc(O)c(CNc2ncnc3cc(C(=O)N4CCCC4)c(Cl)cc23)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.42
PDE5A O76074 2/20 0.38
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
AURKA O14965 3/20 0.35
RPS6KB1 P23443 3/20 0.35
AURKB Q96GD4 2/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
MAPK10 P53779 3/20 0.34
EGFR P00533 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
MAPK8 P45983 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6326778 0.90 CDK1 (0.41) CDK1PDE5AALDH1A1KDM4EMAPK1
SCHEMBL2995398 0.89 CDK1 (0.42) CDK1PDE5AALDH1A1KDM4EMAPK1
SCHEMBL8312247 0.88 CDK1 (0.39) CDK1PDE5AALDH1A1KDM4EMAPK1
SCHEMBL8308640 0.85 CDK1 (0.37) CDK1PDE5AALDH1A1KDM4EMAPK1
SCHEMBL6326818 0.84 CDK1 (0.47) CDK1PDE5AALDH1A1KDM4EMAPK1
Hydrochloric Acid SCHEMBL6322307 0.83 CDK1 (0.46) CDK1PDE5AALDH1A1KDM4EMAPK1
SCHEMBL2991625 0.82 F10 (0.41) CDK1PDE5AALDH1A1AURKARPS6KB1
SCHEMBL8312292 0.81 CDK1 (0.36) CDK1PDE5AALDH1A1MAPK1AURKA
SCHEMBL6322214 0.81 CDK1 (0.39) CDK1PDE5AALDH1A1KDM4EMAPK1
SCHEMBL8308730 0.79 PDE5A (0.36) CDK1PDE5AALDH1A1MAPK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed