SCHEMBL6330737

SCHEMBL6330737

NC(=O)O[C@@H](CO)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
PKM P14618 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
ADRB1 P08588 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2B P41595 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
LMNA P02545 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
EDNRB P24530 1/20 0.44
MAPK1 P28482 1/20 0.44
MC4R P32245 1/20 0.44
CYP2C19 P33261 1/20 0.44
DRD3 P35462 1/20 0.44
MC3R P41968 1/20 0.44
SLC6A3 Q01959 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28500481 1.00 GSR (0.51) GSRCYP1A2CYP2D6PKMSMN1; SMN2
SCHEMBL1043546 1.00 GSR (0.51) GSRCYP1A2CYP2D6PKMSMN1; SMN2
SCHEMBL28552915 0.85 ADRB1 (0.49) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL22813473 0.85 ADRB1 (0.49) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL7511466 0.85 CYP1A2 (0.50) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL21523061 0.85 CYP1A2 (0.50) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL28766159 0.85 CYP1A2 (0.50) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL2836232 0.84 GSR (0.55) GSRCYP1A2CYP2D6PKMSMN1; SMN2
SCHEMBL27811982 0.83 ADRB1 (0.45) ADRB1HTR2AHTR2BSIGMAR1
SCHEMBL514164 0.83 CYP1A2 (0.49) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020240375-A1 IMPROVED PROCESS FOR THE PREPARATION OF ELAGOLIX AND ITS INTERMEDIATES DR. REDDY’S LABORATORIES LIMITED (IN) 2020-12-03 WO disclosed
US-6906066-B2 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2005-06-14 US disclosed
US-20040058960-A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-25 US disclosed
US-20040034063-A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity KO SOO S (US) 2004-02-19 US disclosed
EP-1363881-A2 N-UREIDOALKYL-PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Pharma Company (US) 2003-11-26 EP disclosed
US-6605623-B1 Prevention of asthma and other allergic diseases BRISTOL-MYERS SQUIBB PHARMA CO. 2003-08-12 US disclosed
US-6525069-B1 Such as N-(t-butyl)-N'-(2-((3-(4-fluorophenyl)methyl)piperi -dinyl)methyl)cyclohexyl)urea; prevention of asthma and other allergic diseases BRISTOL-MYERS SQUIBB PHARMA CO. 2003-02-25 US disclosed
WO-2001098269-A2 N-UREIDOALKYL-PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-12-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040058960-A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity CCR3, CCR1, CCR10 GSR 4126/4885CYP1A2 3062/4885CYP2D6 3262/4885
US-20040034063-A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity CCR3, CCR1, CCR10 GSR 4126/4885CYP1A2 3062/4885CYP2D6 3262/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.