SCHEMBL633112

SCHEMBL633112

C#CN1CCN(CCOC)CC1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.38
GBA1 P04062 1/20 0.33
MAP4K4 O95819 1/20 0.32
NPC1 O15118 1/20 0.31
KDM1A O60341 1/20 0.31
PIK3CA P42336 1/20 0.30
MTOR P42345 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8149011 0.82 HSD11B1 (0.47) HSD11B1GBA1MAP4K4NPC1KDM1A
SCHEMBL6057032 0.82
SCHEMBL4893194 0.82 HSD11B1 (0.47) HSD11B1GBA1MAP4K4NPC1KDM1A
SCHEMBL1783124 0.79 HSD11B1 (0.41) HSD11B1GBA1MAP4K4NPC1KDM1A
SCHEMBL18725913 0.76 DRD2 (0.39)
SCHEMBL12125906 0.76 HSD11B1 (0.41) HSD11B1GBA1MAP4K4NPC1KDM1A
SCHEMBL84800 0.75 HSD11B1 (0.43) HSD11B1GBA1NPC1
SCHEMBL21664675 0.73 HSD11B1 (0.42) HSD11B1GBA1TDP1
SCHEMBL793514 0.73 DRD2 (0.44) HSD11B1GBA1NPC1
SCHEMBL10930283 0.73 HSD11B1 (0.42) HSD11B1GBA1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234992-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS LEPTIN RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2012-02-22 EP claimed