SCHEMBL633193

SCHEMBL633193

COc1ccc(CN2C(=O)COc3ccc(N4C[C@@H](CN5CC(NC(=O)OC(C)(C)C)C5)OC4=O)cc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
SIGMAR1 Q99720 17/20 0.42
LMNA P02545 1/20 0.41
F10 P00742 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL633194 1.00 L3MBTL1 (0.43) L3MBTL1SIGMAR1LMNAF10
SCHEMBL633990 0.84 L3MBTL1 (0.51) L3MBTL1SIGMAR1
SCHEMBL633991 0.84 L3MBTL1 (0.51) L3MBTL1SIGMAR1
SCHEMBL633889 0.78 MAPT (0.50) SIGMAR1LMNAF10
SCHEMBL633887 0.78 MAPT (0.50) SIGMAR1LMNAF10
SCHEMBL14994001 0.78 L3MBTL1 (0.44) L3MBTL1SIGMAR1LMNA
SCHEMBL16162364 0.78 L3MBTL1 (0.44) L3MBTL1SIGMAR1LMNA
SCHEMBL634054 0.77 MCHR1 (0.42) L3MBTL1SIGMAR1
SCHEMBL634053 0.77 MCHR1 (0.42) L3MBTL1SIGMAR1
SCHEMBL15875419 0.75 L3MBTL1 (0.57) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9505750-B2 5-aminocyclylmethyl-oxazolidin-2-one derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2016-11-29 US disclosed
EP-2245028-B1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2012-02-22 EP disclosed
US-20110003789-A1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2011-01-06 US disclosed
EP-2245028-A1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2010-11-03 EP disclosed
WO-2009077989-A1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2009-06-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110003789-A1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES CNKSR1, KCNH1, CBR3 L3MBTL1 2851/4885SIGMAR1 28/4885LMNA 1886/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.