SCHEMBL6332913

SCHEMBL6332913

Cc1c(C)n(S(=O)(=O)c2ccc3c(c2)CNCC3)c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PNMT P11086 6/20 0.53
HTR6 P50406 12/20 0.53
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
HTR2C P28335 2/20 0.44
HTR2B P41595 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6336119 0.88 PNMT (0.60) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL6330390 0.81 HTR6 (0.65) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL6166337 0.80 HTR2C (0.59) HTR6HTR2CHTR2B
SCHEMBL6332768 0.80 HTR6 (0.61) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL6331245 0.75 PNMT (0.51) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL6329299 0.75 PNMT (0.51) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL6330346 0.74 HTR6 (0.58) PNMTHTR6
SCHEMBL30159837 0.74 PCSK9 (0.57) HTR6
SCHEMBL26104217 0.74 PCSK9 (0.57) HTR6
SCHEMBL6328762 0.74 HTR6 (0.62) PNMTHTR6ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849644-B2 Isoquinoline derivatives useful in the treatment of CNS disorders SMITHKLINE BEECHAM P.L.C. (GB) 2005-02-01 US claimed