SCHEMBL633403

SCHEMBL633403

CC(C)N(Cc1c[nH]cn1)c1ccc(CN2CCCC2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
HRH3 Q9Y5N1 1/20 0.39
GRIA2 P42262 4/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
LTA4H P09960 1/20 0.36
CYP2D6 P10635 1/20 0.35
S1PR1 P21453 1/20 0.35
PIK3CD O00329 1/20 0.35
KCNH2 Q12809 1/20 0.34
CDC7 O00311 1/20 0.34
PLK4 O00444 1/20 0.34
AURKA O14965 1/20 0.34
MAPK13 O15264 1/20 0.34
PDPK1 O15530 1/20 0.34
DYRK3 O43781 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PAK4 O96013 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL631566 0.85 ACACB (0.44) ACACBL3MBTL1HRH3GRIA2CYP1A2
SCHEMBL8212380 0.79 TAAR1 (0.59)
SCHEMBL2754389 0.76 L3MBTL1 (0.41) ACACBL3MBTL1HRH3CYP1A2CYP2C9
SCHEMBL19668494 0.75 TAAR1 (0.55)
SCHEMBL632031 0.75 ALDH1A1 (0.40) L3MBTL1CYP1A2CYP2C9CYP2D6PARP1
SCHEMBL632308 0.75 TAAR1 (0.49)
SCHEMBL632131 0.73 TAAR1 (0.43) LTA4H
SCHEMBL631757 0.72 TAAR1 (0.39)
SCHEMBL631728 0.72 TAAR1 (0.38) L3MBTL1
SCHEMBL632978 0.72 TAAR1 (0.38) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076497-B1 AMINOMETHYL-4-IMIDAZOLES HOFFMANN LA ROCHE (CH) 2012-02-22 EP disclosed
EP-2076497-A1 AMINOMETHYL-4-IMIDAZOLES F. Hoffmann-Roche AG (CH) 2009-07-08 EP disclosed
WO-2008046757-A1 AMINOMETHYL-4-IMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2008-04-24 WO disclosed