SCHEMBL634733

SCHEMBL634733

CC[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 7/20 0.74
NR3C1 P04150 4/20 0.74
PGR P06401 3/20 0.74
ALDH1A1 P00352 3/20 0.74
ADRA1A P35348 1/20 0.74
HTR2B P41595 1/20 0.74
LMNA P02545 7/20 0.70
SMN1; SMN2 Q16637 5/20 0.70
TSHR P16473 4/20 0.70
CYP2C19 P33261 3/20 0.70
AR P10275 3/20 0.70
MEN1 O00255 2/20 0.70
KMT2A Q03164 2/20 0.70
HIF1A Q16665 2/20 0.70
THRB P10828 1/20 0.70
ESR1 P03372 1/20 0.70
SERPINA6 P08185 6/20 0.68
BLM P54132 4/20 0.68
MAPT P10636 2/20 0.68
ADORA3 P0DMS8 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL571189 1.00 SHBG (0.74) SHBGNR3C1PGRALDH1A1ADRA1A
SCHEMBL3946610 1.00 SHBG (0.74) SHBGNR3C1PGRALDH1A1ADRA1A
Topterone SCHEMBL140769 0.91 SHBG (0.71) SHBGNR3C1PGRALDH1A1ADRA1A
Topterone SCHEMBL11730925 0.91 SHBG (0.71) SHBGNR3C1PGRALDH1A1ADRA1A
Topterone SCHEMBL8846971 0.91 SHBG (0.71) SHBGNR3C1PGRALDH1A1ADRA1A
Topterone SCHEMBL3844149 0.91 SHBG (0.71) SHBGNR3C1PGRALDH1A1ADRA1A
SCHEMBL11728942 0.89 SHBG (0.68) SHBGNR3C1PGRALDH1A1ADRA1A
SCHEMBL10393805 0.89 SHBG (0.68) SHBGNR3C1PGRALDH1A1ADRA1A
SCHEMBL8236612 0.89 SHBG (0.68) SHBGNR3C1PGRALDH1A1ADRA1A
SCHEMBL29437217 0.88 SHBG (0.71) SHBGNR3C1PGRALDH1A1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 380 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104825397-A Controlled release delivery device containing organosol coating ISA ODIDI 2015-08-12 CN claimed
US-20090263476-A1 Composition of Rapid Disintegrating Direct Compression Buccal Tablet PROVIDENT BANK 2009-10-22 US claimed
CN-101453993-A Controlled release delivery device containing organosol coating ISA ODIDI (CA) 2009-06-10 CN claimed
EP-2007360-A1 CONTROLLED RELEASE DELIVERY DEVICE COMPRISING AN ORGANOSOL COAT Odidi, Isa (CA) 2008-12-31 EP claimed
WO-2007112581-A1 CONTROLLED RELEASE DELIVERY DEVICE COMPRISING AN ORGANOSOL COAT ODIDI ISA (CA) 2007-10-11 WO claimed
EP-1560502-A1 ORAL VETERINARY DRUG DELIVERY SYSTEM AND/OR FEED ADDITIVE DELIVERY SYSTEM, PROCESS FOR THE PREPARATION AND USE THEREOF Szoke, Annamaria (HU) 2005-08-10 EP claimed
WO-2004039172-A1 ORAL VETERINARY DRUG DELIVERY SYSTEM AND/OR FEED ADDITIVE DELIVERY SYSTEM, PROCESS FOR THE PREPARATION AND USE THEREOF SZOKE ANNAMARIA (HU) 2004-05-13 WO claimed
US-6004751-A IDENTIFICATION OF A CANDIDATE INHIBITOR SUBSTANCE THAT IS AN ANTAGONIST OF SEBUM FORMATION ARCH DEVELOPMENT CORPORATION (US) 1999-12-21 US claimed
WO-1998008089-A9 IDENTIFICATION OF ACTIVATORS AND INHIBITORS OF SEBUM FORMATION 1998-05-07 WO claimed
WO-1998008089-A1 IDENTIFICATION OF ACTIVATORS AND INHIBITORS OF SEBUM FORMATION ARCH DEVELOPMENT CORPORATION (US) 1998-02-26 WO claimed
US-4542128-A 17α-Pregn-4-ene-3-oxo-21-carboxylic acid esters, process for the preparation thereof, and use thereof as medicinal agents SCHERING AKTIENGESELLSCHAFT (DE) 1985-09-17 US claimed
EP-4714407-A2 DEVICES TO PROVIDE HANDS FREE SCLERAL DEPRESSION DURING OPHTHALMIC PROCEDURES Alcon Inc. (CH) 2026-03-25 EP disclosed
EP-3157408-B1 DEVICES TO PROVIDE HANDS FREE SCLERAL DEPRESSION DURING OPHTHALMIC PROCEDURES ALCON INC (CH) 2026-03-25 EP disclosed
EP-3432940-B1 COMPLEX BRAIDED SCAFFOLDS FOR IMPROVED TISSUE REGENERATION BIOREZ INC (US) 2025-11-05 EP disclosed
US-20250281509-A1 SEQUENTIAL HORMONE THERAPY TO IMPROVE SURVIVAL AND ENHANCE RESPONSE TO IMMUNE THERAPY IN MEN WITH PROSTATE CANCER THE JOHNS HOPKINS UNIVERSTY 2025-09-11 US disclosed
US-4170518-A Microbiological conversion of sterol derivatives to 5-androsten-17-one derivatives and their use SCHERING AKTIENGESELLSCHAFT (DE) 1979-10-09 US disclosed
US-4160027-A OXYTOCICS, 4A,5A-EPOXY-2A-CYANO-3-OXOSTEROIDES, STEROIDO(2,3-O)ISOOXAZOLES STERLING DRUG INC. (US) 1979-07-03 US disclosed
US-4039669-A DERMATOLOGICAL CONDITIONS, ACNE, STEROIDS STERLING DRUG INC. (US) 1977-08-02 US disclosed
US-3956316-A PROGESTATIONAL AND SALT-RETAINING AGENTS HOFFMANN-LA ROCHE INC. (US) 1976-05-11 US disclosed
US-3944064-A Self-monitored device for releasing agent at functional rate ALZA CORPORATION (US) 1976-03-16 US disclosed