SCHEMBL63495

SCHEMBL63495

CN(C(=O)OCc1ccccc1)C(C#N)C1CCC(CO[Si](C)(C)C(C)(C)C)C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
CTSL P07711 4/20 0.35
CTSB P07858 4/20 0.35
CTSS P25774 4/20 0.35
CTSK P43235 3/20 0.35
ABCB1 P08183 2/20 0.35
PTGIR P43119 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CYP3A4 P08684 2/20 0.33
TSHR P16473 1/20 0.33
CCR5 P51681 5/20 0.33
CCNK O75909 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CDK12 Q9NYV4 1/20 0.33
BTN3A1 O00481 1/20 0.33
CSNK1A1 P48729 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL63843 0.85 PTGIR (0.38) ITGB3ITGA2BCTSLCTSBCTSS
SCHEMBL52324 0.84 ITGB3 (0.41) ITGB3ITGA2BCTSLCTSBCTSS
SCHEMBL2633971 0.83
SCHEMBL31045282 0.72 SIGMAR1 (0.51) ABCB1SIGMAR1CYP3A4TSHRBTN3A1
SCHEMBL52346 0.70 JAK2 (0.32) CTSLCTSBCTSSCTSKCYP3A4
SCHEMBL1118425 0.70 SIGMAR1 (0.42) ITGB3ITGA2BCTSLCTSBCTSS
SCHEMBL17352069 0.70 ITGB3 (0.44) ITGB3ITGA2BCTSLCTSBCTSS
SCHEMBL63846 0.68 ITGB3 (0.42) ITGB3ITGA2BCTSLCTSBCTSS
SCHEMBL4972692 0.67 ABCB1 (0.38) ITGB3ITGA2BCTSLCTSBCTSS
SCHEMBL1117736 0.67 DPP4 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129398-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-06 US disclosed
US-20090253677-A1 HIV Integrase Inhibitors BRISTOL-MYERS SQUIBB COMPANY 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090253677-A1 HIV Integrase Inhibitors DNTT, POLB, UNG ITGB3 2078/4885ITGA2B 1968/4885CTSL 3453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.