SCHEMBL6349873

SCHEMBL6349873

CCCOc1ccc(-c2ccc3c(c2)C=C(C(=O)OC)CCN3C=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.39
CCR5 P51681 7/20 0.37
PLA2G2A P14555 1/20 0.37
ALDH1A1 P00352 4/20 0.37
HPGD P15428 3/20 0.37
GAA P10253 3/20 0.37
MAPK1 P28482 2/20 0.37
TSHR P16473 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GLA P06280 1/20 0.37
THRB P10828 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
RUNX1 Q01196 1/20 0.37
ATM Q13315 1/20 0.37
CBFB Q13951 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ABCB1 P08183 2/20 0.37
ALPL P05186 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6351503 0.92 ALDH1A1 (0.43) ERN1CCR5ALDH1A1HPGDGAA
SCHEMBL6350067 0.92 CCR5 (0.45) CCR5PLA2G2ATSHRABCB1ALPL
SCHEMBL6351904 0.92 CCR5 (0.39) CCR5ALDH1A1HPGDGAACCR7
SCHEMBL6342973 0.91 CCR5 (0.38) CCR5ALDH1A1HPGDGAAALPL
SCHEMBL6349978 0.90 MPL (0.39) ERN1CCR5ALDH1A1HPGDGAA
SCHEMBL6351996 0.90 CCR5 (0.33) CCR5ALDH1A1HPGDGAAKDM4E
SCHEMBL6341329 0.89 CCR5 (0.38) CCR5HPGDCCR7CCR2MAPT
SCHEMBL3458669 0.86 CCR5 (0.49) CCR5ALPLCCR7CCR2MAPT
SCHEMBL3458663 0.86 CCR5 (0.49) CCR5ALPLCCR7CCR2MAPT
SCHEMBL6341045 0.83 MEN1 (0.43) CCR5PLA2G2AALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed