SCHEMBL6350449

SCHEMBL6350449

CCCN(CCCC(=O)O)c1ccc(Br)cc1C=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH3A1 P30838 3/20 0.46
ALDH1A3 P47895 3/20 0.46
ALDH1A1 P00352 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.42
ERN1 O75460 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
HCAR3 P49019 1/20 0.36
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
GLA P06280 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34
CYSLTR2 Q9NS75 1/20 0.33
CYSLTR1 Q9Y271 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3458716 0.96 ALDH1A1 (0.45) ALDH3A1ALDH1A3ALDH1A1PTGDR2ERN1
SCHEMBL7541512 0.95 PTGDR2 (0.42) ALDH3A1ALDH1A3ALDH1A1PTGDR2ERN1
SCHEMBL7543270 0.86 ALDH1A1 (0.45) ALDH3A1ALDH1A3ALDH1A1PTGDR2ERN1
SCHEMBL6517350 0.85 PTGDR2 (0.40) ALDH3A1ALDH1A3ALDH1A1PTGDR2ERN1
SCHEMBL7541400 0.84 PTGDR2 (0.46) ALDH1A1PTGDR2ERN1KMT2AMEN1
SCHEMBL7544691 0.84 PTGDR2 (0.41) ALDH1A1PTGDR2ERN1KMT2AMEN1
SCHEMBL7487895 0.84 ALDH3A1 (0.41) ALDH3A1ALDH1A3ALDH1A1PTGDR2ERN1
SCHEMBL3458964 0.83 ALDH3A1 (0.42) ALDH3A1ALDH1A3ALDH1A1PTGDR2ERN1
SCHEMBL7684624 0.83 PTGDR2 (0.45) ALDH1A1PTGDR2ERN1KMT2AMEN1
SCHEMBL3157614 0.82 PTGDR2 (0.40) ALDH1A3ALDH1A1PTGDR2ERN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1211239-A1 PROCESS FOR THE PREPARATION OF 2,3-DIHYDROAZEPINE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2002-06-05 EP disclosed