SCHEMBL6367132

SCHEMBL6367132

O=C(c1ccc(F)cc1)c1ccc(C[C@H](NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc(Cl)cc(Cl)c2)C(=O)O)cc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.66
ITGB1 P05556 14/20 0.66
ITGB7 P26010 6/20 0.66
ITGAV P06756 2/20 0.55
ITGA5 P08648 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368398 0.96 ITGA4 (0.69) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL5687080 0.93 ITGA4 (0.66) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6372387 0.93 ITGA4 (0.66) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6367900 0.91 ITGA4 (0.63) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6372412 0.89 ITGA4 (0.72) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6368166 0.88 ITGB1 (0.72) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6368456 0.87 ITGA4 (0.70) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6368512 0.87 ITGA4 (0.72) ITGA4ITGB1ITGB7ITGA5
SCHEMBL6367880 0.87 ITGA4 (0.69) ITGA4ITGB1ITGB7ITGAVITGA5
SCHEMBL6368438 0.87 ITGA4 (0.69) ITGA4ITGB1ITGB7ITGAVITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP disclosed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US disclosed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP disclosed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO disclosed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed