SCHEMBL6367902

SCHEMBL6367902

O=C(O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.59
ITGA5 P08648 4/20 0.59
ITGA4 P13612 6/20 0.57
POLB P06746 1/20 0.56
ITGB7 P26010 3/20 0.54
ITGAV P06756 5/20 0.53
HCRTR1 O43613 1/20 0.48
HCRTR2 O43614 1/20 0.48
ITGA2 P17301 1/20 0.47
KCNQ1 P51787 1/20 0.46
BRD4 O60885 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL630186 0.91 ITGB1 (0.56) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL630187 0.91 ITGB1 (0.56) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL6368195 0.90 ITGB1 (0.64) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL5172120 0.89 ITGB1 (0.55) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL630086 0.88 POLB (0.56) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL630087 0.88 POLB (0.56) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL6368166 0.88 ITGB1 (0.72) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL629837 0.88 KCNQ1 (0.62) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL630658 0.88 ITGB1 (0.53) ITGB1ITGA5ITGA4POLBITGB7
SCHEMBL629838 0.88 KCNQ1 (0.62) ITGB1ITGA5ITGA4POLBITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed