SCHEMBL6375358

SCHEMBL6375358

O=C(O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cc(Cl)c(Cl)s1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.53
ITGA4 P13612 10/20 0.53
ITGA5 P08648 3/20 0.52
ITGB7 P26010 2/20 0.51
ITGAV P06756 6/20 0.46
ITGA2 P17301 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368978 0.92 ITGB1 (0.52) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL6368403 0.86 ITGB1 (0.50) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL6368457 0.85 ITGA4 (0.48) ITGB1ITGA4ITGA5ITGB7CA1
SCHEMBL6368648 0.83 ITGB1 (0.50) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL6368456 0.83 ITGA4 (0.70) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL23519443 0.81 ITGB1 (0.75) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL23499865 0.81 ITGB1 (0.75) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL23519426 0.81 ITGB1 (0.75) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL23519669 0.81 ITGB1 (0.75) ITGB1ITGA4ITGA5ITGB7ITGAV
SCHEMBL23499866 0.81 ITGB1 (0.75) ITGB1ITGA4ITGA5ITGB7ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed