SCHEMBL6368648

SCHEMBL6368648

O=C(O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cc(Br)c(Cl)s1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.50
ITGA5 P08648 3/20 0.50
ITGA4 P13612 8/20 0.49
ITGB7 P26010 3/20 0.49
ITGAV P06756 6/20 0.49
MMP8 P22894 1/20 0.42
MMP12 P39900 1/20 0.42
MMP13 P45452 1/20 0.42
ITGA2 P17301 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368978 0.91 ITGB1 (0.52) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6374007 0.87 ITGB1 (0.51) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6374041 0.86 MMP8 (0.60) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6375358 0.83 ITGB1 (0.53) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6368403 0.82 ITGB1 (0.50) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6368398 0.82 ITGA4 (0.69) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6373924 0.80 ITGB1 (0.59) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6368166 0.80 ITGB1 (0.72) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6372387 0.80 ITGA4 (0.66) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL5687080 0.80 ITGA4 (0.66) ITGB1ITGA5ITGA4ITGB7ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed