SCHEMBL6375377

SCHEMBL6375377

COc1ccc(C(=O)N(CC(=O)N2CCN(CCc3ccncc3)CC2)c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.62
THRB P10828 4/20 0.51
SIGMAR1 Q99720 1/20 0.50
ACHE P22303 1/20 0.47
DRD3 P35462 1/20 0.47
CHRM3 P20309 1/20 0.47
DRD2 P14416 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
SLC2A1 P11166 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6295711 0.99 POLB (0.61) POLBTHRBSIGMAR1ACHEDRD3
Hydrochloric Acid SCHEMBL4840396 0.99 POLB (0.61) POLBTHRBSIGMAR1ACHEDRD3
Hydrochloric Acid SCHEMBL6219381 0.94 SIGMAR1 (0.57) POLBTHRBSIGMAR1ACHEDRD3
SCHEMBL4837431 0.93 SIGMAR1 (0.57) POLBSIGMAR1ACHEDRD3CHRM3
SCHEMBL4832532 0.91 ACHE (0.58) POLBSIGMAR1ACHECHRM3
SCHEMBL6191181 0.88 POLB (0.59) POLBTHRBSIGMAR1DRD3DRD2
Hydrochloric Acid SCHEMBL4836733 0.88 POLB (0.60) POLBTHRB
SCHEMBL4839910 0.86 TP53 (0.55) POLBTHRBSIGMAR1ACHEDRD3
Hydrochloric Acid SCHEMBL4832406 0.84 POLB (0.58) POLBTHRBSIGMAR1DRD3DRD2
SCHEMBL4842118 0.83 ACHE (0.66) POLBSIGMAR1ACHECHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005023422-A2 PRODUCTION AND USE OF IONIC LIQUIDS CONTAINING THIOCYANATO ANIONS SOLVENT INNOVATION GMBH (DE) 2005-03-17 WO disclosed
US-6855715-B1 Serine protease inhibitors ELI LILLY AND COMPANY (US) 2005-02-15 US disclosed
EP-1192135-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2002-04-03 EP disclosed
EP-1192132-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2002-04-03 EP disclosed
WO-2000076970-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2000-12-21 WO disclosed
WO-2000076971-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2000-12-21 WO disclosed