SCHEMBL6376540

SCHEMBL6376540

CC(C)(C)OC(=O)N(CCc1ccccc1)Cc1cc(C(=O)O)ccc1N

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
LPAR1 Q92633 8/20 0.43
LPAR5 Q9H1C0 8/20 0.43
HDAC6 Q9UBN7 1/20 0.42
RCE1 Q9Y256 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6378379 0.92 SLC7A5 (0.43) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL6378384 0.85 ALDH1A1 (0.48) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL6377823 0.85 ALDH1A1 (0.48) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL8326453 0.85 CDC25B (0.37) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL6655287 0.85 SLC7A5 (0.45) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL6947602 0.84 PTGER4 (0.43) HDAC1HDAC3HDAC2NCOR2HDAC6
SCHEMBL6383755 0.83 MEN1 (0.48) HDAC1LPAR1LPAR5HDAC6RCE1
SCHEMBL27334618 0.81 ALDH1A1 (0.41) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL8326411 0.81 LPAR1 (0.38) HDAC1HDAC3HDAC2NCOR2LPAR1
SCHEMBL9823156 0.80 HDAC1 (0.54) HDAC1HDAC3HDAC2NCOR2LPAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1225895-B1 FAB I INHIBITORS AFFINIUM PHARM INC (CA) 2005-05-04 EP disclosed
US-6762201-B1 SUCH AS N-((2-AMINO-5-(N-METHYL-N-((1-METHYLINDOL-2-YL) -METHYL)CARBAMOYL)PHENYL)METHYL)-N-METHYLACETAMIDE; BACTERIAL INFECTIONS AFFINIUM PHARMACEUTICALS, INC. (CA) 2004-07-13 US disclosed