SCHEMBL8326411

SCHEMBL8326411

CC(C)(C)OC(=O)N(Cc1cc(C(=O)O)ccc1N)CC(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 6/20 0.38
LPAR5 Q9H1C0 6/20 0.38
CDC25B P30305 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PLA2G2D Q9UNK4 1/20 0.34
THRB P10828 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
GFER P55789 1/20 0.34
PLEC Q15149 1/20 0.34
AAK1 Q2M2I8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327800 0.91 ALOX15 (0.38) HDAC3HDAC1HDAC2NCOR2SSTR4
SCHEMBL8327876 0.84 POLB (0.44) ALDH1A1
SCHEMBL8327873 0.84 POLB (0.44) ALDH1A1
SCHEMBL8326453 0.83 CDC25B (0.37) LPAR1LPAR5CDC25BHDAC3HDAC1
SCHEMBL6947602 0.82 PTGER4 (0.43) CDC25BHDAC3HDAC1HDAC2NCOR2
SCHEMBL28609267 0.82 HDAC3 (0.38) CDC25BHDAC3HDAC1HDAC2NCOR2
SCHEMBL6941296 0.82 CDC25B (0.42) CDC25BHDAC3HDAC1HDAC2NCOR2
SCHEMBL6376540 0.81 HDAC1 (0.43) LPAR1LPAR5HDAC3HDAC1HDAC2
SCHEMBL7425320 0.76 KDM4E (0.38) CDC25BHDAC3KDM4EALDH1A1GAA
SCHEMBL8326945 0.75 KMT2A (0.40) ALDH1A1MAPTTHRBHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed