SCHEMBL6378153

SCHEMBL6378153

COc1ccc(Cc2nc(C)ccc2OS(=O)(=O)C(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
PDE10A Q9Y233 2/20 0.39
LTA4H P09960 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE2A O00408 3/20 0.35
MDM4 O15151 1/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
HTT P42858 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17440325 0.80 KDM4E (0.43) ALDH1A1KDM4ETP53ATM
SCHEMBL6377285 0.76 KDM4E (0.49) ALDH1A1RAB9AKDM4EHPGDSMN1; SMN2
SCHEMBL6378210 0.73 KDM4E (0.73) ALDH1A1RAB9AKDM4EHPGDPDE3B
SCHEMBL18188355 0.73 S1PR4 (0.38) RAB9AKDM4ESMN1; SMN2NPC1
SCHEMBL4061114 0.72 S1PR4 (0.39) KDM4EL3MBTL1
SCHEMBL1997269 0.72 CA1 (0.57)
SCHEMBL608235 0.72 TACR1 (0.33) KDM4E
SCHEMBL7043778 0.71 MTNR1A (0.45) ALDH1A1LTA4HSMN1; SMN2TP53HTT
SCHEMBL15492954 0.71 CA1 (0.32)
Hydrogen Sulfide SCHEMBL5082548 0.70 CA1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100334085-C Quinuclidine compound and medicine containing the same as active ingredient EISAI R & D CO LTD (JP) 2007-08-29 CN disclosed
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
CN-1377349-A Quinuclidine compound and medicine containing the same as active ingredient EISAI CO LTD (JP) 2002-10-30 CN disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed