SCHEMBL6378783

SCHEMBL6378783

COc1ncccc1Cc1cccs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP1A2 P05177 3/20 0.42
CYP2D6 P10635 3/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
KDM1A O60341 3/20 0.40
SLC13A5 Q86YT5 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP2C9 P11712 2/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
TSHR P16473 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9390272 0.77 PIK3CD (0.43) ALDH1A1CYP2C9TSHRADRA1DHTR6
SCHEMBL6376093 0.76 KDM1A (0.50) CYP3A4KDM1ASLC13A5MAOAMAOB
SCHEMBL235980 0.76 POLB (0.54) L3MBTL1CYP3A4KDM1ASLC13A5MAOA
SCHEMBL2203168 0.76 POLB (0.54) L3MBTL1CYP3A4KDM1ASLC13A5MAOA
SCHEMBL6379419 0.75 CYP2C9 (0.37) L3MBTL1ALDH1A1CYP2C9TSHRMEN1
SCHEMBL91503 0.73 SLC13A5 (0.50) RAB9ANPC1L3MBTL1KDM1ASLC13A5
SCHEMBL6047280 0.73 KDM1A (0.54) CYP3A4CYP2C19KDM1ASLC13A5MAOA
SCHEMBL30505689 0.72 CYP2C9 (0.50) RAB9ANPC1CYP1A2CYP2D6CYP3A4
SCHEMBL5382166 0.72 LTA4H (0.55) RAB9ANPC1ALDH1A1CYP2C9MEN1
SCHEMBL27585504 0.72 KDM1A (0.41) L3MBTL1CYP3A4KDM1ASLC13A5MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed