SCHEMBL6380294

SCHEMBL6380294

COc1cc2nccc(Oc3ccc(N)cc3F)c2cc1OC.COc1cc2nccc(Oc3ccc(NC(=O)Nc4cc(C)no4)cc3F)c2cc1OC

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 12/20 0.64
PDGFRA P16234 2/20 0.62
KDR P35968 2/20 0.57
MET P08581 6/20 0.57
AXL P30530 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5653628 0.95 FLT3 (0.70) FLT3PDGFRAKDRMETAXL
SCHEMBL5652832 0.85 KDR (0.65) FLT3PDGFRAKDRMET
SCHEMBL6376965 0.82 FLT3 (0.79) FLT3PDGFRAKDRMETAXL
Hydrochloric Acid SCHEMBL5653983 0.81 FLT3 (0.78) FLT3PDGFRAKDRMETAXL
SCHEMBL6380290 0.81 FLT3 (0.54) FLT3PDGFRAKDRMETAXL
SCHEMBL5652690 0.80 FLT3 (0.76) FLT3PDGFRAKDRMETAXL
SCHEMBL5653905 0.79 KDR (0.74) FLT3PDGFRAKDRMETAXL
SCHEMBL20434905 0.78 FLT3 (1.00) FLT3
SCHEMBL166914 0.78 AXL (0.67) PDGFRAKDRMETAXL
SCHEMBL698529 0.78 AXL (0.66) FLT3PDGFRAKDRMETAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1382604-B1 QUINOLINE DERIVATIVE HAVING AZOLYL GROUP AND QUINAZOLINE DERIVATIVE KIRIN BREWERY (JP) 2005-12-28 EP disclosed
EP-1382604-A1 QUINOLINE DERIVATIVE HAVING AZOLYL GROUP AND QUINAZOLINE DERIVATIVE KIRIN BEER KABUSHIKI KAISHA (JP) 2004-01-21 EP disclosed