SCHEMBL6401547

SCHEMBL6401547

O=C(COc1ccc(O)c(O)c1)N(Cc1cccs1)c1cccnc1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 14/20 0.75
TP53 P04637 5/20 0.53
LMNA P02545 3/20 0.50
THRB P10828 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6408147 0.87 TRPM8 (0.72) TRPM8TP53LMNATHRBTDP1
SCHEMBL2717456 0.86 TRPM8 (0.82) TRPM8TP53LMNATDP1POLB
SCHEMBL2720078 0.86 TRPM8 (0.85) TRPM8TP53LMNATHRBTDP1
SCHEMBL2717987 0.86 TRPM8 (0.81) TRPM8TP53LMNATDP1POLB
SCHEMBL2718358 0.86 TRPM8 (1.00) TRPM8TP53
SCHEMBL30582820 0.85 TRPM8 (0.71) TRPM8TP53LMNATHRBTDP1
SCHEMBL30582849 0.85 TRPM8 (0.74) TRPM8TP53LMNATHRBPOLB
SCHEMBL2719236 0.85 TRPM8 (0.80) TRPM8TP53LMNATHRB
SCHEMBL2717851 0.85 TRPM8 (0.74) TRPM8TP53LMNATHRBPOLB
SCHEMBL2717537 0.85 TRPM8 (0.71) TRPM8TP53LMNATHRBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061698-A9 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 SENOMYX, INC. (US) 2012-09-13 WO disclosed
WO-2012061698-A2 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 SENOMYX, INC. (US) 2012-05-10 WO disclosed