SCHEMBL6402817

SCHEMBL6402817

Cc1ccc(S(=O)(=O)N(C)CC(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.58
TP53 P04637 2/20 0.57
MAPT P10636 1/20 0.57
GAA P10253 3/20 0.56
KDM4E B2RXH2 2/20 0.52
LMNA P02545 2/20 0.52
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
ADRB2 P07550 1/20 0.51
TDP1 Q9NUW8 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CNR2 P34972 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA3 P07451 1/20 0.49
CA4 P22748 1/20 0.49
CA6 P23280 1/20 0.49
CA5A P35218 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5899682 0.87 GAA (0.50) KMT2AMAPTGAARAB9AADRB2
SCHEMBL5899593 0.87 KMT2A (0.54) KMT2AMAPTGAAADRB2TDP1
SCHEMBL11603483 0.85 RECQL (0.59) KMT2AKDM4ELMNARAB9ANPC1
SCHEMBL27628054 0.85 TDP1 (0.49) KMT2AMAPTGAAADRB2TDP1
SCHEMBL5899425 0.85 ALDH1A1 (0.56) KMT2AMAPTGAAKDM4ELMNA
SCHEMBL5899473 0.84 GAA (0.50) KMT2AMAPTGAAADRB2TDP1
SCHEMBL2335204 0.82 GAA (0.56) KMT2AMAPTGAARAB9AADRB2
SCHEMBL6320992 0.80 POLB (0.55) KMT2AMAPTGAAKDM4ELMNA
SCHEMBL5899493 0.80 GAA (0.48) KMT2AMAPTGAAADRB2TDP1
SCHEMBL11579297 0.79 POLB (0.64) KMT2AMAPTGAAKDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1501830-A1 7-ARYL-3,9-DIAZABICYCLO[3.3.1]NON-6-ENE DERIVATIVES AND THEIR USE AS RENIN INHIBITORS IN THE TREATMENT OF HYPERTENSION, CARDIOVASCULAR OR RENAL DISEASES Actelion Pharmaceuticals Ltd. (CH) 2005-02-02 EP disclosed
WO-2003093267-A1 7-ARYL-3,9-DIAZABICYCLO(3.3.1)NON-6-ENE DERIVATIVES AND THEIR USE AS RENIN INHIBITORS IN THE TREATMENT OF HYPERTENSION, CARDIOVASCULAR OR RENAL DISEASES ACTELION PHARMACEUTICALS LTD (CH) 2003-11-13 WO disclosed