SCHEMBL6403014

SCHEMBL6403014

COc1ccc2c(c1)C[C@@H](O)CC2

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.66
DRD3 P35462 6/20 0.66
DRD4 P21917 2/20 0.58
MTNR1A P48039 1/20 0.58
MTNR1B P49286 1/20 0.58
CA1 P00915 4/20 0.55
CA2 P00918 4/20 0.55
ACHE P22303 4/20 0.55
CYP19A1 P11511 2/20 0.52
CYP26A1 O43174 1/20 0.49
HTR1A P08908 1/20 0.45
SIGMAR1 Q99720 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629692 1.00 DRD2 (0.66) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL4001498 1.00 DRD2 (0.66) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL7958191 0.93 DRD2 (0.58) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL8765765 0.90 DRD2 (0.58) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL4000913 0.90 DRD2 (0.58) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL4000915 0.90 DRD2 (0.58) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL23343811 0.85 DRD2 (0.54) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL3961628 0.85 DRD2 (0.54) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL8983525 0.81 DRD2 (0.68) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL10977596 0.80 DRD2 (0.68) DRD2DRD3DRD4MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050153408-A1 7-substituted-2-tetralone or bisulfite adduct is reduced microorganism (Candida) to optically active 7-substituted-2-tetralol;sulfonyl group is introduced to hydroxy group to form optically active 7-substituted-2-sulfonyloxytetralin; nitrogen substituent is introduced via ammonia; industrial scale KANEKA CORPORATION (JP) 2005-07-14 US disclosed
EP-1457570-A1 PROCESS FOR PREPARATION OF 2-AMINOTETRALIN DERIVATIVES AND INTERMEDIATES THEREOF KANEKA CORPORATION (JP) 2004-09-15 EP disclosed