SCHEMBL6404849

SCHEMBL6404849

COc1ccc2c(c1)C[C@@H](NCCc1ccccc1)CC2

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.76
KMT2A Q03164 1/20 0.76
GRIN2B Q13224 11/20 0.74
GRIN1 Q05586 2/20 0.74
DRD2 P14416 2/20 0.71
DRD3 P35462 2/20 0.71
SIGMAR1 Q99720 1/20 0.57
MTNR1A P48039 1/20 0.54
MTNR1B P49286 1/20 0.54
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
ACHE P22303 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6404851 1.00 POLB (0.76) POLBKMT2AGRIN2BGRIN1DRD2
SCHEMBL388869 0.88 POLB (0.65) POLBKMT2AGRIN2BGRIN1DRD2
SCHEMBL355042 0.88 DRD2 (0.67) POLBKMT2AGRIN2BGRIN1DRD2
SCHEMBL9516292 0.88 DRD2 (0.67) POLBKMT2AGRIN2BGRIN1DRD2
SCHEMBL9515249 0.88 DRD2 (0.67) POLBKMT2AGRIN2BGRIN1DRD2
Hydrochloric Acid SCHEMBL9305508 0.86 DRD2 (0.65) POLBKMT2AGRIN2BGRIN1DRD2
Hydrochloric Acid SCHEMBL8767433 0.86 DRD2 (0.65) POLBKMT2AGRIN2BGRIN1DRD2
Hydrochloric Acid SCHEMBL9304463 0.86 DRD2 (0.65) POLBKMT2AGRIN2BGRIN1DRD2
Hydrochloric Acid SCHEMBL7326528 0.85 POLB (0.97) POLBKMT2AGRIN2BGRIN1DRD2
Hydrochloric Acid SCHEMBL7335860 0.84 POLB (0.74) POLBKMT2AGRIN2BGRIN1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050153408-A1 7-substituted-2-tetralone or bisulfite adduct is reduced microorganism (Candida) to optically active 7-substituted-2-tetralol;sulfonyl group is introduced to hydroxy group to form optically active 7-substituted-2-sulfonyloxytetralin; nitrogen substituent is introduced via ammonia; industrial scale KANEKA CORPORATION (JP) 2005-07-14 US disclosed
EP-1457570-A1 PROCESS FOR PREPARATION OF 2-AMINOTETRALIN DERIVATIVES AND INTERMEDIATES THEREOF KANEKA CORPORATION (JP) 2004-09-15 EP disclosed