SCHEMBL6405616

SCHEMBL6405616

COc1ccc2c(c1)C[C@H](OS(C)(=O)=O)CC2

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.57
DRD3 P35462 6/20 0.57
CA1 P00915 4/20 0.53
CA2 P00918 4/20 0.53
ACHE P22303 4/20 0.53
MTNR1A P48039 3/20 0.52
MTNR1B P49286 2/20 0.52
DRD4 P21917 2/20 0.49
CYP19A1 P11511 2/20 0.47
HTR2C P28335 1/20 0.43
CYP26A1 O43174 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
THRB P10828 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958716 0.94 CA1 (0.53) DRD2DRD3CA1CA2ACHE
SCHEMBL8766020 0.92 DRD2 (0.51) DRD2DRD3CA1CA2ACHE
SCHEMBL5485492 0.83 DRD2 (0.66) DRD2DRD3CA1CA2ACHE
SCHEMBL6951811 0.82 HTR1D (0.39) DRD2DRD3CA1CA2ACHE
SCHEMBL6958304 0.82 HTR1D (0.39) DRD2DRD3CA1CA2ACHE
SCHEMBL6951816 0.82 HTR1D (0.39) DRD2DRD3CA1CA2ACHE
SCHEMBL6401807 0.81 DRD2 (0.50) DRD2DRD3CA1CA2ACHE
SCHEMBL4857120 0.80 CA1 (0.45) CA1CA2MTNR1AMTNR1BHTR2C
SCHEMBL6953263 0.80 CA1 (0.45) CA1CA2MTNR1AMTNR1BHTR2C
SCHEMBL629488 0.78 MTNR1A (0.61) DRD2DRD3CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050153408-A1 7-substituted-2-tetralone or bisulfite adduct is reduced microorganism (Candida) to optically active 7-substituted-2-tetralol;sulfonyl group is introduced to hydroxy group to form optically active 7-substituted-2-sulfonyloxytetralin; nitrogen substituent is introduced via ammonia; industrial scale KANEKA CORPORATION (JP) 2005-07-14 US disclosed
EP-1457570-A1 PROCESS FOR PREPARATION OF 2-AMINOTETRALIN DERIVATIVES AND INTERMEDIATES THEREOF KANEKA CORPORATION (JP) 2004-09-15 EP disclosed