SCHEMBL6405846

SCHEMBL6405846

CCCc1c(OCCCN2C(=O)CSC2=O)ccc2c(CC(C)(C)C)onc12

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 12/20 0.64
NR1H3 Q13133 10/20 0.64
ALDH1A1 P00352 1/20 0.36
GRM2 Q14416 1/20 0.36
PPARA Q07869 7/20 0.34
PPARD Q03181 7/20 0.34
PPARG P37231 6/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6404754 0.88 NR1H2 (0.48) NR1H2NR1H3GRM2PPARAPPARD
SCHEMBL6408328 0.85 NR1H2 (0.46) NR1H2NR1H3GRM2PPARAPPARD
SCHEMBL6405354 0.85 NR1H2 (0.72) NR1H2NR1H3PPARAPPARDPPARG
SCHEMBL6097922 0.84 NR1H2 (0.74) NR1H2NR1H3GRM2PPARAPPARD
SCHEMBL6405513 0.83 NR1H2 (0.44) NR1H2NR1H3GRM2PPARAPPARD
SCHEMBL6407458 0.81 NR1H2 (0.41) NR1H2NR1H3ALDH1A1GRM2PPARA
SCHEMBL6100435 0.78 NR1H2 (1.00) NR1H2NR1H3PPARAPPARDPPARG
SCHEMBL6411684 0.77 NR1H2 (0.57) NR1H2NR1H3ALDH1A1
SCHEMBL6405323 0.72 NR1H2 (0.55) NR1H2NR1H3PPARAPPARDPPARG
SCHEMBL1595776 0.72 NR1H2 (0.71) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534696-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS Merck & Co., Inc. (US) 2005-06-01 EP claimed
WO-2004011448-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS MERCK & CO., INC. (US) 2004-02-05 WO claimed
EP-1534696-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS Merck & Co., Inc. (US) 2005-06-01 EP disclosed
WO-2004011448-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS MERCK & CO., INC. (US) 2004-02-05 WO disclosed