SCHEMBL6408049

SCHEMBL6408049

COc1ccc(C(=O)NCc2cc(C(=O)Nc3ccccc3)no2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.55
RAB9A P51151 6/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
KCNK9 Q9NPC2 1/20 0.54
KMT2A Q03164 6/20 0.53
MEN1 O00255 5/20 0.53
MAPT P10636 4/20 0.53
HSD17B10 Q99714 3/20 0.53
TSHR P16473 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
KDM4E B2RXH2 2/20 0.52
ALDH1A1 P00352 4/20 0.51
ADORA3 P0DMS8 1/20 0.51
MAPK1 P28482 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
POLB P06746 1/20 0.50
CTDSP1 Q9GZU7 1/20 0.50
ATM Q13315 1/20 0.49
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6408618 0.94 SMN1; SMN2 (0.62) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6402547 0.90 SMN1; SMN2 (0.57) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6407778 0.90 HSD17B10 (0.62) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6405915 0.89 NPC1 (0.64) NPC1RAB9ASMN1; SMN2KCNK9KMT2A
SCHEMBL6404235 0.89 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6402278 0.88 HDAC6 (0.57) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL6410111 0.88 SMN1; SMN2 (0.62) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6410519 0.87 NPC1 (0.59) NPC1RAB9ASMN1; SMN2MAPTHSD17B10
SCHEMBL6405888 0.86 SMN1; SMN2 (0.53) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6402541 0.86 RXFP1 (0.65) NPC1RAB9ASMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528737-B Novel heteroaryl carboxamides HOFFMANN LA ROCHE 2012-07-04 CN disclosed
US-20050171358-A1 Substituted isoxazole alkylamine derivative and agri-and horticultural fungicide SDS BIOTECH K.K. (JP) 2005-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171358-A1 Substituted isoxazole alkylamine derivative and agri-and horticultural fungicide AHR, ERG28, CYP1A2 NPC1 1915/4885RAB9A 4044/4885SMN1; SMN2 4458/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.