SCHEMBL6409124

SCHEMBL6409124

CC(C)C(=O)N[C@@H](CCN1CCC2(CC1)CCN(Cc1ccccn1)C2=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.43
EGLN1 Q9GZT9 2/20 0.43
HCRTR2 O43614 1/20 0.41
ALDH1A1 P00352 2/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
SLC5A7 Q9GZV3 1/20 0.39
CTRB1 P17538 1/20 0.39
PPARG P37231 1/20 0.38
GPR88 Q9GZN0 1/20 0.38
CACNA1G O43497 1/20 0.37
CACNA1H O95180 1/20 0.37
CACNA1I Q9P0X4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6409962 0.87 ROCK2 (0.46) CCR5ROCK2ROCK1KDM4EGPR88
Hydrochloric Acid SCHEMBL6415642 0.86 CCR5 (0.46) CCR5ALDH1A1ROCK2ROCK1
SCHEMBL6409016 0.84 HCRTR2 (0.43) CCR5HCRTR2ALDH1A1ROCK2ROCK1
SCHEMBL6409501 0.84 HCRTR2 (0.43) CCR5HCRTR2ALDH1A1ROCK2ROCK1
Hydrochloric Acid SCHEMBL6410988 0.84 HCRTR2 (0.42) CCR5HCRTR2ALDH1A1ROCK2ROCK1
SCHEMBL6409300 0.83 CCR5 (0.44) CCR5ROCK2ROCK1LMNA
SCHEMBL6409295 0.83 CCR5 (0.44) CCR5ROCK2ROCK1LMNA
Hydrochloric Acid SCHEMBL6410911 0.83 UTS2R (0.46) CCR5
SCHEMBL6412938 0.83 EGLN1 (0.52) EGLN1HCRTR2ALDH1A1KDM4ELMNA
SCHEMBL6414757 0.82 CCR5 (0.45) CCR5ALDH1A1ROCK2ROCK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050075326-A1 Spiro compounds and methods for the modulation of chemokine receptor activity VIROCHEM PHARMA INC (CA) 2005-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075326-A1 Spiro compounds and methods for the modulation of chemokine receptor activity CXCR1, CXCR4, CXCR2 CCR5 4/4885EGLN1 2490/4885HCRTR2 247/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.